Regioselective 2-acylation of N-substituted pyrroles by intramolecular delivery

Browse by...

Deposit

Highlights

More informations

Title		Regioselective 2-acylation of N-substituted pyrroles by intramolecular delivery
Authors		Jefford, Charles Tang, Qian Boukouvalas, John
Published in		Tetrahedron letters. 1990, vol. 31, no. 7, p. 995-998
Abstract		N-substituted pyrroles prepared from α-amino acids are converted to their mixed anhydrides by treatment with an acid chloride and base. Subsequent treatment with AlCl3 brings about rearrangement to the corresponding 2-acyl derivatives in overall yields of 55-81%.
Identifiers		DOI: 10.1016/S0040-4039(00)94412-5
Full text		Article (Published version) (1.8 MB) - Limited access to UNIGE Other version: https://linkinghub.elsevier.com/retrieve/pii/S0040403900944125
Structures		Faculté des sciences / Section de chimie et biochimie / Département de chimie organique
Project		Swiss National Science Foundation: 20-5380.87
Citation (ISO format)		JEFFORD, Charles, TANG, Qian, BOUKOUVALAS, John. Regioselective 2-acylation of N-substituted pyrroles by intramolecular delivery. In: Tetrahedron Letters, 1990, vol. 31, n° 7, p. 995-998. doi: 10.1016/S0040-4039(00)94412-5 https://archive-ouverte.unige.ch/unige:152799