Controlled Iontophoretic Delivery in Vitro and in Vivo of ARN14140-A Multitarget Compound for Alzheimer's Disease
Contributeurs/tricesSinghal, Mayank; Merino, Virginia; Rosini, Michela; Cavalli, Andrea; Kalia, Yogeshvar
Publié dansMolecular Pharmaceutics, vol. 16, no. 8, p. 3460-3468
Date de publication2019
Résumé
Mots-clés
- Administration, Cutaneous
- Alzheimer Disease/drug therapy
- Animals
- Biological Availability
- Brain/metabolism
- Drug Stability
- Feasibility Studies
- Galantamine/administration & dosage/pharmacokinetics
- Heterocyclic Compounds, 4 or More Rings/administration & dosage/pharmacology
- Humans
- Iontophoresis
- Male
- Memantine/administration & dosage/pharmacokinetics
- Nootropic Agents/administration & dosage/pharmacokinetics
- Permeability
- Rats
- Rats, Wistar
- Skin/metabolism
- Skin Absorption
- Swine
- Tissue Distribution
Structure d'affiliation
Citation (format ISO)
SINGHAL, Mayank et al. Controlled Iontophoretic Delivery in Vitro and in Vivo of ARN14140-A Multitarget Compound for Alzheimer’s Disease. In: Molecular Pharmaceutics, 2019, vol. 16, n° 8, p. 3460–3468. doi: 10.1021/acs.molpharmaceut.9b00252
Fichiers principaux (1)
Article (Published version)
Identifiants
- PID : unige:138467
- DOI : 10.1021/acs.molpharmaceut.9b00252
- PMID : 31241959
ISSN du journal1543-8384