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| Enhancing Oral Delivery of Biologics: A Non-Competitive and Cross-Reactive Anti-Leptin Receptor Nanofitin Demonstrates a Gut-Crossing Capacity in an Ex Vivo Porcine Intestinal Model | Pharmaceutics |  | | 2024 | 128 | 262 |
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| Effects of a diverse prebiotic fibre supplement on HbA1c, insulin sensitivity and inflammatory biomarkers in pre-diabetes: a pilot placebo-controlled randomised clinical trial | British journal of nutrition |  | | 2024 | 1 | 0 |
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| Compound K14 inhibits bacterial killing and protease activity in Dictyostelium discoideum phagosomes | PloS one |  | | 2024 | 59 | 190 |
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| Targeted Nanofitin-drug Conjugates Achieve Efficient Tumor Delivery and Therapeutic Effect in an EGFRpos Mouse Xenograft Model | Molecular cancer therapeutics |  | | 2023 | 77 | 211 |
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| CEMIP ( HYBID , KIAA1199 ): structure, function and expression in health and disease | The FEBS journal |  | | 2022 | 188 | 350 |
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| 5-ethyl-2’-deoxyuridine fragilizes Klebsiella pneumoniae outer wall and facilitates intracellular killing by phagocytic cells | PloS one |  | | 2022 | 89 | 172 |
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| Chemoenzymatic synthesis of original stilbene dimers possessing wnt inhibition activity in triple-negative breast cancer cells using the enzymatic secretome of Botrytis cinerea pers | Frontiers in chemistry |  | | 2022 | 241 | 222 |
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| Using protease inhibitors to improve protein stability in the presence of skin: A case study on the stability of insulin like growth factor 1 | European journal of pharmaceutics and biopharmaceutics |  | | 2021 | 1 | 0 |
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| Functional and anatomical characterization of atrophic age-related macular degeneration in an aged mouse model | Journal of Ophthalmology and Research |  | | 2021 | 465 | 392 |
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| Heat-stability study of various insulin types in tropical temperature conditions: new insights towards improving diabetes care | PLOS ONE |  | | 2021 | 396 | 525 |
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| Novel Mechanism for an Old Drug: Phenazopyridine is a Kinase Inhibitor Affecting Autophagy and Cellular Differentiation | Frontiers in pharmacology |  | | 2021 | 154 | 351 |
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| From Conception to Development: Investigating PROTACs Features for Improved Cell Permeability and Successful Protein Degradation | Frontiers in Chemistry |  | | 2021 | 510 | 1,158 |
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| Platelet Transforming Growth Factor-β1 Induces Liver Sinusoidal Endothelial Cells to Secrete Interleukin-6 | Cells |  | | 2020 | 370 | 211 |
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| Identification of anti-mycobacterium and anti-legionella compounds with potential distinctive structural scaffolds from an HD-PBL using phenotypic screens in amoebae host models | Frontiers in Microbiology |  | | 2020 | 332 | 233 |
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| Cooperative binding of the tandem WW domains of PLEKHA7 to PDZD11 promotes conformation-dependent interaction with tetraspanin 33 | Journal of Biological Chemistry |  | | 2020 | 303 | 217 |
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| Drug repurposing in oncology: Compounds, pathways, phenotypes and computational approaches for colorectal cancer | Biochimica et Biophysica Acta. Reviews on Cancer |  | | 2019 | 494 | 1,606 |
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| Tamoxifen prolongs survival and alleviates symptoms in mice with fatal X-linked myotubular myopathy | Nature Communications |  | | 2018 | 516 | 376 |
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| Modeling and resistant alleles explain the selectivity of antimalarial compound 49c towards apicomplexan aspartyl proteases | EMBO Journal |  | | 2018 | 684 | 15 |
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| Mammalian RAD52 Functions in Break-Induced Replication Repair of Collapsed DNA Replication Forks | Molecular cell |  | | 2016 | 71 | 212 |
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| In silico driven design and synthesis of rhodanine derivatives as novel antibacterials targeting the enoyl reductase InhA | Journal of medicinal chemistry |  | | 2016 | 680 | 6 |
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| Differences in Conformational Dynamics between Plasmodium falciparum and Human Hsp90 Orthologues Enable the Structure-Based Discovery of Pathogen-Selective Inhibitors | Journal of medicinal chemistry |  | | 2014 | 724 | 796 |
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| Diapocynin, a Dimer of the NADPH Oxidase Inhibitor Apocynin, Reduces ROS Production and Prevents Force Loss in Eccentrically Contracting Dystrophic Muscle | PloS one |  | | 2014 | 634 | 653 |
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| Analysis of the cross-reactivity and of the 1.5 A crystal structure of the Malassezia sympodialis Mala s 6 allergen, a member of the cyclophilin pan-allergen family | Biochemical journal |  | | 2006 | 503 | 0 |
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| Structural Insights into the ATP Binding Pocket of the Anaplastic Lymphoma Kinase by Site-Directed Mutagenesis, Inhibitor Binding Analysis, and Homology Modeling | Journal of medicinal chemistry |  | | 2006 | 138 | 0 |
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| Inhibition of Plasmodium falciparum Fatty Acid Biosynthesis: Evaluation of FabG, FabZ, and FabI as Drug Targets for Flavonoids | Journal of medicinal chemistry |  | | 2006 | 198 | 1 |
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| Recombinant expression and biochemical characterization of the unique elongating β-Ketoacyl-acyl carrier protein synthase involved in fatty acid biosynthesis of Plasmodium falciparum using natural and artificial substrates | The Journal of biological chemistry |  | | 2006 | 171 | 132 |
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| Abl inhibitor BMS354825 binding mode in Abelson kinase revealed by molecular docking studies | Leukemia |  | | 2005 | 128 | 0 |
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| Unique substrate specificity of anaplastic lymphoma kinase (ALK): development of phosphoacceptor peptides for the assay of ALK activity | Biochemistry |  | | 2005 | 564 | 0 |
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