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HDM-PAMPA to predict gastrointestinal absorption, binding percentage, equilibrium and kinetics constants with human serum albumin and using 2 end-point measurements Bujard, Alban; Petit, Charlotte; Carrupt, Pierre-Alain; Rudaz, Serge; Schappler, Julie 2017
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Passive Intestinal Absorption of Representative Plant Secondary Metabolites: A Physicochemical Study Petit, Charlotte; Ceccarelli, Martina; Cretton, Sylvian; Houriet, Joëlle; ... Wolfender, Jean-Luc 2017
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Prediction of the Passive Intestinal Absorption of Medicinal Plant Extract Constituents with the Parallel Artificial Membrane Permeability Assay (PAMPA) Petit, Charlotte; Bujard, Alban; Skalicka-Woźniak, Krystyna; Cretton, Sylvian; ... Wolfender, Jean-Luc 2016
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Normal phase HPLC-based activity profiling of non-polar crude plant extracts - acetylcholinesterase inhibiting guttiferones from Montrouziera cauliflora as a case study Landreau, Anne; Bertrand, Samuel; Simoes-Pires, Claudia; Marcourt, Laurence; ... Wolfender, Jean-Luc 2016
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Modification of a PAMPA model to predict passive gastrointestinal absorption and plasma protein binding Bujard, Alban; Voirol, Hervé; Carrupt, Pierre-Alain; Schappler, Julie 2015
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Inhibition screening method of microsomal UGTs using the cocktail approach Gradinaru, Julieta; Romand, Stéphanie Anne; Geiser, Laurent; Carrupt, Pierre-Alain; ... Rudaz, Serge 2015
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cIEF for rapid pKa determination of small molecules: A proof of concept Romand, Stéphanie Anne; Schappler, Julie; Veuthey, Jean-Luc; Carrupt, Pierre-Alain; Martel, Sophie 2014
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Predicting both passive intestinal absorption and the dissociation constant toward albumin using the PAMPA technique Bujard, Alban; Sol, Marine; Carrupt, Pierre-Alain; Martel, Sophie 2014
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Computational Studies on Sirtuins from Trypanosoma cruzi: Structures, Conformations and Interactions with Phytochemicals Sacconnay, Lionel; Angleviel, Mélissa; Randazzo, Giuseppe Marco; Ferreira Queiroz, Marcos Marcal; ... Nurisso, Alessandra 2014
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Isolation and biological activity of compounds from Garcinia preussii Biloa Messi, Bernadette; Ho, Raimana; Meli Lannang, Alain; Cressend, Delphine; ... Cuendet, Muriel 2014
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Antifungals and acetylcholinesterase inhibitors from the stem bark of Croton heliotropiifolius Ferreira Queiroz, Marcos Marcal; Ferreira Queiroz, Emerson; Zeraik, Maria Luiza; Marti, Guillaume; ... Wolfender, Jean-Luc 2014
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Aurones as histone deacetylase inhibitors: identification of key features Zwick, Vincent; Chatzivasileiou, Alkiviadis-Orfefs; Deschamps, Nathalie; Roussaki, Marina; ... Cuendet, Muriel 2014
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Large, chemically diverse dataset of logP measurements for benchmarking studies Martel, Sophie; Gillerat, Fabrice; Carosati, E.; Maiarelli, D.; ... Carrupt, Pierre-Alain 2013
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Unsymmetrical binding modes of HOPNO inhibitor of tyrosinase: From model complexes to the enzyme Bochot, C.; Favre, Anne Elisabeth; Dubois, C.; Baptiste, B.; ... Jamet, H. 2013
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High performance affinity chromatography (HPAC) as a high-throughput screening tool in drug discovery to study drug–plasma protein interactions Vuignier, Karine; Guillarme, Davy; Veuthey, Jean-Luc; Carrupt, Pierre-Alain; Schappler, Julie 2013
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Analytical Strategy to Characterize Drug–Plasma Interactions: From High Throughput to In-depth Analysis Vuignier, Karine; Veuthey, Jean-Luc; Carrupt, Pierre-Alain; Schappler, Julie 2013
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Global analytical strategy to measure drug–plasma protein interactions: from high-throughput to in-depth analysis Vuignier, Karine; Veuthey, Jean-Luc; Carrupt, Pierre-Alain; Schappler, Julie 2013
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New high throughput screening method for drug release measurements Pelczarska, Aleksandra Paulina; Delie Salmon, Florence; Domańska, Urszula; Carrupt, Pierre-Alain; Martel, Sophie 2013
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Comparison of various silica-based monoliths for the analysis of large biomolecules Vuignier, Karine; Fekete, Szabolcs; Carrupt, Pierre-Alain; Veuthey, Jean-Luc; Guillarme, Davy 2013
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Anti-inflammatory, antimicrobial and antioxidant activities of Diospyros bipindensis (Gürke) extracts and its main constituents Cesari, Ilaria; Hoerle, Mélanie; Simoes Avello, Claudia; Grisoli, P.; ... Brusotti, G. 2013
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HDAC6 as a target for neurodegenerative diseases: what makes it different from the other HDACs? Simoes Avello, Claudia; Zwick, Vincent; Nurisso, Alessandra; Schenker, Esther; ... Cuendet, Muriel 2013
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Synthesis physicochemical profile and PAMPA study of new NO-donor edaravone co-drugs Rolando, Barbara; Filieri, Andrea; Chegaev, Konstantin; Lazzarato, Loretta; ... Gasco, Alberto 2012
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Antioxidant potential and radical scavenging effects of flavonoids from the leaves of Psidium cattleianum grown in French Polynesia Ho, Raimana; Aude, Violette; Cressend, Delphine; Raharivelomanana, Phila; ... Hostettmann, Kurt 2012
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Characterization of drug-protein interactions by capillary electrophoresis hyphenated to mass spectrometry Vuignier, Karine; Veuthey, Jean-Luc; Carrupt, Pierre-Alain; Schappler, Julie 2012
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Ultra High Pressure Liquid Chromatography for Crude Plant Extract Profiling Eugster, Philippe; Guillarme, Davy; Rudaz, Serge; Veuthey, Jean-Luc; ... Wolfender, Jean-Luc 2011
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Biarylmethoxy isonipecotanilides as potent and selctive inhibitors of blood coagulation facture Xa Lopoplo, G.; Fiorella, F.; de Candia, M.; Nicoletti, O.; ... Altomare, C. 2011
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In vitro blood brain barrier models as a screening tool for colloidal drug delivery systems and other nanosystems Garcel, Aude; Martel, Sophie; Carrupt, Pierre-Alain; Doelker, Eric; Delie Salmon, Florence 2010
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The permeability P-glycoprotein: a focus on enantioselectivity and brain distribution Choong, Eva; Dobrinas, Maria; Carrupt, Pierre-Alain; Eap, Chin Bin 2010
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Stereoselective block of hERG channel by bupivacaine scrutinized at molecular level Sintra Grilo, Liliana; Carrupt, Pierre-Alain; Daina, Antoine 2010
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Improvement of a capillary electrophoresis/frontal analysis (CE/FA) method for determining binding constants: Discussion on relevant parameters Vuignier, Karine; Schappler, Julie; Veuthey, Jean-Luc; Carrupt, Pierre-Alain; Martel, Sophie 2010
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Physicochemical profile and in vitro permeation behavior of a new class of non-steroidal anti-inflammatory drug candidates Rolando, B.; Lazzarato, L.; Di Stilo, A.; Fruttero, Roberta; ... Gasco, Alberto 2010
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Entacapone and tolcapone, two catechol O-methyltransferase inhibitors, block fibril formation of alpha-synuclein and beta-amyloid and protect against amyloid-induced toxicity Di Giovanni, S.; Eleuteri, S.; Paleologou, K. E.; Yin, G.; ... Lashuel, H. A. 2010
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Molecular electrocatalysis for oxygen reduction by cobalt porphyrins adsorbed at liquid/liquid interfaces Su, B.; Hatay, I.; Trojanek, A.; Samec, Z.; ... Girault, Hubert 2010
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Stereoselective inhibition of the hERG1 potassium channel Sintra Grilo, Liliana; Carrupt, Pierre-Alain; Abriel, Hugues 2010
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Standard machine learning algorithms applied to UPLC-TOF/MS metabolic fingerprinting for the discovery of wound biomarkers in Arabidopsis thaliana Boccard, Julien; Kalousis, Alexandros; Hilario, Mélanie; Lantéri, Pierre; ... Rudaz, Serge 2010
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Drug-protein binding: a critical review of analytical tools Vuignier, Karine; Schappler, Julie; Veuthey, Jean-Luc; Carrupt, Pierre-Alain; Martel, Sophie 2010
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Advances in LC platforms for drug discovery Nicoli, Raul; Martel, Sophie; Rudaz, Serge; Wolfender, Jean-Luc; ... Guillarme, Davy 2010
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High-throughput log P determination by MEEKC coupled with UV and MS detections Henchoz, Yveline; Romand, Stéphanie; Schappler, Julie; Rudaz, Serge; ... Carrupt, Pierre-Alain 2010
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Antioxidant profiling of new chemical entities from synthetic and natural origin Cressend, Delphine; Reist, Marianne; Carrupt, Pierre-Alain 2009
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Olive phenols efficiently inhibit the oxidation of serum albumin-bound linoleic acid and butyrylcholine esterase Roche, Marjolaine; Dufour, Claire; Loonis, Michèle; Reist, Marianne; ... Dangles, Olivier 2009
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Metabolite profiling of plant extracts by ultra-high-pressure liquid chromatography at elevated temperature coupled to time-of-flight mass spectrometry Grata, Elia; Guillarme, Davy; Glauser, Gaétan; Boccard, Julien; ... Wolfender, Jean-Luc 2009
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Monoamine oxidase inhibition by Rhodiola rosea L. roots Van Diermen, Daphné; Marston, Andrew; Bravo, Juan; Reist, Marianne; ... Hostettmann, Kurt 2009
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In silico tools and in vitro HTS approaches to determine lipophilicity during the drug discovery process Martel, Sophie; Gasparik, Vincent; Carrupt, Pierre-Alain 2009
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Breast cancer resistance protein (BCRP/ABCG2): new inhibitors and QSAR studies by a 3D linear solvation energy approach Nicolle, Edwige; Boccard, Julien; Guilet, David; Dijoux-Franca, Marie-Geneviève; ... Boumendjel, Ahcène 2009
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Lipophilicity of basic drugs measured by hydrophilic interaction chromatography Bard, Bruno; Carrupt, Pierre-Alain; Martel, Sophie 2009
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A 3D linear solvation energy model to quantify the affinity of flavonoid derivatives toward P-glycoprotein Boccard, Julien; Bajot, Fania; Di Pietro, Attilio; Rudaz, Serge; ... Carrupt, Pierre-Alain 2009
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QSAR analysis and molecular modeling of ABCG2-specific inhibitors Nicolle, Edwige; Boumendjel, A.; Macalou, S.; Genoux, E.; ... Di Pietro, A. 2009
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Edaravone derivatives containing NO-donor functions Chegaev, Konstantin; Cena, Clara; Giorgis, Marta; Rolando, Barbara; ... Gasco, Alberto 2009
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A fast screening strategy for characterizing peptide delivery by transdermal iontophoresis Henchoz, Yveline; Abla, Nada; Veuthey, Jean-Luc; Carrupt, Pierre-Alain 2009
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Rapid log P determination of natural products in crude plant extracts from UHPLC-TOF-MS profiling data - an additional parameter for dereplication and bioavailability Eugster, Philippe; Martel, Sophie; Guillarme, Davy; Carrupt, Pierre-Alain; Wolfender, Jean-Luc 2009
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