| Title | Authors / Editors | Date |
unige:92508 |
HDM-PAMPA to predict gastrointestinal absorption, binding percentage, equilibrium and kinetics constants with human serum albumin and using 2 end-point measurements |
Bujard, Alban; Petit, Charlotte; Carrupt, Pierre-Alain; Rudaz, Serge; Schappler, Julie |
2017 |
unige:101913 |
ERE-dependent transcription and cell proliferation: Independency of these two processes mediated by the introduction of a sulfone function into the weak estrogen estrothiazine |
Jacquot, Yves; Spaggiari, Dany; Schappler, Julie; Lesniewska, Eric; ... Leclercq, Guy |
2017 |
unige:78263 |
Modification of a PAMPA model to predict passive gastrointestinal absorption and plasma protein binding |
Bujard, Alban; Voirol, Hervé; Carrupt, Pierre-Alain; Schappler, Julie |
2015 |
unige:88245 |
Inhibition screening method of microsomal UGTs using the cocktail approach |
Gradinaru, Julieta; Romand, Stéphanie Anne; Geiser, Laurent; Carrupt, Pierre-Alain; ... Rudaz, Serge |
2015 |
unige:40568 |
cIEF for rapid pKa determination of small molecules: A proof of concept |
Romand, Stéphanie Anne; Schappler, Julie; Veuthey, Jean-Luc; Carrupt, Pierre-Alain; Martel, Sophie |
2014 |
unige:46356 |
Predicting both passive intestinal absorption and the dissociation constant toward albumin using the PAMPA technique |
Bujard, Alban; Sol, Marine; Carrupt, Pierre-Alain; Martel, Sophie |
2014 |
unige:28608 |
Large, chemically diverse dataset of logP measurements for benchmarking studies |
Martel, Sophie; Gillerat, Fabrice; Carosati, E.; Maiarelli, D.; ... Carrupt, Pierre-Alain |
2013 |
unige:17531 |
Biarylmethoxy isonipecotanilides as potent and selctive inhibitors of blood coagulation facture Xa |
Lopoplo, G.; Fiorella, F.; de Candia, M.; Nicoletti, O.; ... Altomare, C. |
2011 |
unige:10644 |
Physicochemical profile and in vitro permeation behavior of a new class of non-steroidal anti-inflammatory drug candidates |
Rolando, B.; Lazzarato, L.; Di Stilo, A.; Fruttero, Roberta; ... Gasco, Alberto |
2010 |
unige:22796 |
Comparing metoclopramide electrotransport kinetics in vitro and in vivo |
Cazares Delgadillo, Jennyfer; Benaziza, Ines; Balaguer-Fernández, Cristina; Calatayud-Pascual, Aracely; ... Kalia, Yogeshvar |
2010 |
unige:22914 |
Using transdermal iontophoresis to increase granisetron delivery across skin in vitro and in vivo: effect of experimental conditions and a comparison with other enhancement strategies |
Cazares Delgadillo, Jennyfer; Ganem-Rondero, Adriana; Quintanar-Guerrero, David; López-Castellano, Alicia C; ... Kalia, Yogeshvar |
2010 |
unige:19744 |
Nanomedicines for active targeting: physico-chemical characterization of paclitaxel-loaded anti-HER2 immunonanoparticles and in vitro functional studies on target cells |
Cirstoiu, Adriana; Buchegger, Franz; Bossy, Leila; Kosinski, M; ... Delie Salmon, Florence |
2009 |
unige:1205 |
Localization and quantification of biodegradable particles in an intestinal cell model: the influence of particle size |
Gaumet, Marie; Gurny, Robert; Delie Salmon, Florence |
2009 |
unige:3979 |
Breast cancer resistance protein (BCRP/ABCG2): new inhibitors and QSAR studies by a 3D linear solvation energy approach |
Nicolle, Edwige; Boccard, Julien; Guilet, David; Dijoux-Franca, Marie-Geneviève; ... Boumendjel, Ahcène |
2009 |
unige:3983 |
A 3D linear solvation energy model to quantify the affinity of flavonoid derivatives toward P-glycoprotein |
Boccard, Julien; Bajot, Fania; Di Pietro, Attilio; Rudaz, Serge; ... Carrupt, Pierre-Alain |
2009 |
unige:4067 |
In vitro screening assays to identify natural or synthetic acetylcholinesterase inhibitors: thin layer chromatography versus microplate methods |
Di Giovanni, Saviana; Borloz, Aline; Urbain, Aurélie; Marston, Andrew; ... Reist, Marianne |
2008 |
unige:4068 |
High throughput UV method for the estimation of thermodynamic solubility and the determination of the solubility in biorelevant media |
Bard, Bruno; Martel, Sophie; Carrupt, Pierre-Alain |
2008 |
unige:4081 |
The PAMPA technique as a HTS tool for partition coefficients determination in different solvent/water systems |
Ottaviani, Giorgio; Martel, Sophie; Escarala, Caroline; Nicolle, Edwige; Carrupt, Pierre-Alain |
2008 |
unige:10651 |
Structure-permeation relationships for the non-invasive transdermal delivery of cationic peptides by iontophoresis |
Schuetz, Yannic; Carrupt, Pierre-Alain; Naik, Aarti; Guy, Richard H.; Kalia, Yogeshvar |
2006 |
unige:22643 |
Effect of amino acid sequence on transdermal iontophoretic peptide delivery |
Schuetz, Yannic; Naik, Aarti; Guy, Richard H.; Kalia, Yogeshvar |
2005 |