Human recombinant monoamine oxidase B as reliable and efficient enzyme source for inhibitor screening
Contributeurs/tricesNovaroli, L.; Reist, Marianne; Favre, Elisabeth; Carotti, Angelo; Catto, M.; Carrupt, Pierre-Alain
Publié dansBioorganic & medicinal chemistry, vol. 13, no. 22, p. 6212-6217
Date de publication2005
Résumé
Mots-clés
- Blood Platelets/drug effects/enzymology
- Coumarins/analysis/chemistry/pharmacology
- Drug Evaluation, Preclinical/methods
- Humans
- Inhibitory Concentration 50
- Monoamine Oxidase/*drug effects/*genetics/metabolism
- Monoamine Oxidase Inhibitors/analysis/chemistry/*pharmacology
- Pyridazines/analysis/classification/pharmacology
- Recombinant Proteins/*genetics
Structure d'affiliation
Citation (format ISO)
NOVAROLI, L. et al. Human recombinant monoamine oxidase B as reliable and efficient enzyme source for inhibitor screening. In: Bioorganic & medicinal chemistry, 2005, vol. 13, n° 22, p. 6212–6217. doi: 10.1016/j.bmc.2005.06.043
Fichiers principaux (1)
Article
Identifiants
- PID : unige:10616
- DOI : 10.1016/j.bmc.2005.06.043
- PMID : 16054369
ISSN du journal0968-0896